Spirooxindoles as novel 3D-fragment scaffolds: Synthesis and screening against CYP121 from M. tuberculosis

Fragment-Based Approaches to the Development of Mycobacterium tuberculosis CYP121 Inhibitors

Natural product-inspired fragment-based drug discovery: Development of M. tuberculosis CYP121 inhibitors

Fragment-based drug discovery of potent and selective CYP121 inhibitors for tuberculosis

CHAPTER 8 Fragment-Based Discovery of Antibacterials

ChemInform Abstract: Regioselective Conversion of Arenes to N‐Aryl‐1,2,3‐triazoles Using C—H Borylation.

Understanding "On-Water" Catalysis of Organic Reactions. Effects of H⁺ and Li⁺ Ions in the Aqueous Phase and Nonreacting Competitor H-Bond Acceptors in the Organic Phase: On H₂O versus on D₂O for Huisgen Cycloadditions

Small-molecule inhibitors that target protein-protein interactions in the RAD51 family of recombinases

Regioselective conversion of arenes to N-aryl-1,2,3-triazoles using C-H borylation.

Overcoming the Limitations of Fragment Merging: Rescuing a Strained Merged Fragment Series Targeting Mycobacterium tuberculosis CYP121