Publications
Substrate Fragmentation for the Design of M.tuberculosis CYP121 Inhibitors
ChemMedChem
(2016)
11
1924
(doi: 10.1002/cmdc.201600248)
Spirooxindoles as novel 3D-fragment scaffolds: Synthesis and screening against CYP121 from M. tuberculosis
Bioorg Med Chem Lett
(2016)
26
3735
(doi: 10.1016/j.bmcl.2016.05.073)
Fragment-Based Approaches to the Development of Mycobacterium tuberculosis CYP121 Inhibitors.
Journal of medicinal chemistry
(2016)
59
3272
(doi: 10.1021/acs.jmedchem.6b00007)
ChemInform Abstract: Regioselective Conversion of Arenes to N‐Aryl‐1,2,3‐triazoles Using C—H Borylation.
ChemInform
(2015)
46
no
(doi: 10.1002/chin.201510175)
Understanding “On-Water” Catalysis of Organic Reactions. Effects of H+ and Li+ Ions in the Aqueous Phase and Nonreacting Competitor H-Bond Acceptors in the Organic Phase: On H2O versus on D2O for Huisgen Cycloadditions
J Org Chem
(2015)
80
1809
(doi: 10.1021/jo502732y)
Natural product-inspired fragment-based drug discovery: Development of M. tuberculosis CYP121 inhibitors
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY
(2015)
250
Fragment-based drug discovery of potent and selective CYP121 inhibitors for tuberculosis
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY
(2015)
250
Small-Molecule Inhibitors That Target Protein-Protein Interactions in the RAD51 Family of Recombinases
ChemMedChem
(2014)
10
296
(doi: 10.1002/cmdc.201402428)
Regioselective conversion of arenes to N-aryl-1,2,3-triazoles Using C-H Borylation
Chemistry (Weinheim an der Bergstrasse, Germany)
(2014)
20
11680
(doi: 10.1002/chem.201403021)
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