Publications
Overcoming the limitations of fragment merging: rescuing a strained merged fragment series targeting Mycobacterium tuberculosis CYP121.
ChemMedChem
(2013)
8
1451
(doi: 10.1002/cmdc.201300219)
Water and organic synthesis: A focus on the in-water and on-water border. Reversal of the in-water breslow hydrophobic enhancement of the normal endo -effect on crossing to on-water conditions for huisgen cycloadditions with increasingly insoluble organic liquid and solid 2π-dipolarophiles
The Journal of Organic Chemistry
(2013)
78
3276
(doi: 10.1021/jo400055g)
Fragment-Based Approaches in Drug Discovery and Chemical Biology
Biochemistry
(2012)
51
4990
(doi: 10.1021/bi3005126)
ChemInform Abstract: Asymmetric Electrocyclic Reactions
ChemInform
(2011)
42
no
(doi: 10.1002/chin.201149243)
Fragment based approach to targeting the Rad51:BRCA2 protein-protein interaction
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY
(2011)
242
Trapping of palindromic ligands within native transthyretin prevents amyloid formation.
Proceedings of the National Academy of Sciences
(2010)
107
20483
(doi: 10.1073/pnas.1008255107)
Water: Nature's reaction enforcer-comparative effects for organic synthesis "in-water" and "on-water"
Chem Rev
(2010)
110
6302
(doi: 10.1021/cr100162c)
ChemInform Abstract: Regioselectivity and endo/exo Selectivity in the Cycloadditions of the Phthalazinium Dicyanomethanide 1,3‐Dipole with Unsymmetrical Alkene and Alkyne Dipolarophiles. Unexpected Reversals of Regiochemistry: A Combined Experimental and DFT Theoretical Study.
ChemInform
(2010)
32
no
(doi: 10.1002/chin.200143032)
ChemInform Abstract: Ligand Design for Intermolecular Asymmetric Mizoroki—Heck Reactions
ChemInform
(2010)
41
no
(doi: 10.1002/chin.201020231)
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