Publications
Allosteric targeting of aurora a kinase using small molecules: A step forward towards next generation medicines?
Current Medicinal Chemistry
(2019)
26
2234
Development of inhibitors against Mycobacterium abscessus tRNA (m1G37) methyltransferase (TrmD) using fragment-based approaches.
J Med Chem
(2019)
62
7210
(doi: 10.1021/acs.jmedchem.9b00809)
Structure-guided fragmentbased drug discovery at the synchrotron: Screening binding sites and correlations with hotspot mapping
Philosophical Transactions of the Royal Society A Mathematical Physical and Engineering Sciences
(2019)
377
20180422
(doi: 10.1098/rsta.2018.0422)
Development of Inhibitors Against Mycobacterium Abscessus tRNA (m1G37) Methyltransferase (TrmD) Using Fragment-Based Approaches
(2019)
(doi: 10.26434/chemrxiv.8131847)
meta‐Nitration of Arenes Bearing ortho/para Directing Group(s) Using C−H Borylation
Chemistry – A European Journal
(2019)
25
8018
(doi: 10.1002/chem.201901633)
Fragment-based discovery of a new class of inhibitors targeting mycobacterial tRNA modification
(2019)
(doi: 10.1101/564013)
Fragment-Based Approach to Targeting Inosine-5'-monophosphate Dehydrogenase (IMPDH) from Mycobacterium tuberculosis.
J Med Chem
(2018)
61
2806
(doi: 10.1021/acs.jmedchem.7b01622)
Mass spectrometry for fragment screening.
Essays in Biochemistry
(2017)
61
465
(doi: 10.1042/ebc20170071)
Effect of DMSO on Protein Structure and Interactions Assessed by Collision-Induced Dissociation and Unfolding.
Anal Chem
(2017)
89
9976
(doi: 10.1021/acs.analchem.7b02329)
Fragment Screening against the EthR–DNA Interaction by Native Mass Spectrometry
Angewandte Chemie (International ed. in English)
(2017)
56
7488
(doi: 10.1002/anie.201702888)
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